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BDPC (systematic name 4-(4-bromophenyl)-4-(dimethylamino)-1-(2-phenylethyl)cyclohexanol; also known as bromadol) is a potent narcotic analgesic with a distinctive arylcyclohexylamine chemical structure. It was developed by Daniel Lednicer at Upjohn in the 1970s. Initial studies estimated that it was around 10,000 times the strength of morphine in animal models. However, later studies using more modern techniques assigned a value of 504 times the potency of morphine for the more active trans-isomer. 

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To date, it is unknown if this drug (BDPC) has been used by humans, however, it was seized along with three kilograms of acetylfentanyl in an April 25, 2013 police action in Montreal, Canada, and has reportedly continued to be available on the designer drug black market internationally. Analogues where the para-bromine is replaced by chlorine or CH3 retain similar activity, as does the meta-hydroxy derivative. 

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Compound trans-4-(p-bromophenyl)-4-(dimethylamino)-1-(2-thiophen-2-yl-ethyl)-cyclohexanol (C8813), structurally unrelated to morphine, ((BDPC) is a novel analgesic. The present study examined the antinociception, opioid receptor selectivity and in vitro activity of C8813. The antinociceptive activity was evaluated using mouse hot plate and acetic acid writhing tests.  

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Bromadol (3), also referred to as BDPC (trans-4-(p-bromophenyl)-4-(dimethylamino)-1-phenethylcyclohexanol), was among the most potent and efficacious compounds studied here. Using a standard mouse hot plate assay, Liu et al. (2003). previously suggested that the analgesic potency of bromadol may be around 2.9 times that of fentanyl (Sharma et al. 2019). The herein reported in vitro potencies for βarr2 and mini-Gi recruitment echo this, as the EC 50 values for bromadol were 7.6-and 10.8-fold lower than those obtained for fentanyl using the same respective assays 

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However, as discussed further, it remains difficult to directly compare in vivo analgesic potency to in vitro potency values. Interestingly, the in vivo antinociceptive potency reported by Liu et al. (2003) was greater than what may be expected based on opioid receptor binding affinity data (Sharma et al. 2019). Although determination of binding affinity was outside the scope of the current study, the high in vitro efficacy and potency at MOR reported here may provide an explanation for this. BDPC 

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It was originally stated that BDPC/bromadol had 10,000 times the analgesic potency of morphine in animal studies although a more recent study, comparing analgesic potency using a standard mouse hot plate assay where BDPC/bromadol was introduced by intraperitoneal injection, suggests that its analgesic potency may be lower, at around 500 times that of morphine and 2.9 times that of fentanyl. 

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Other Names: CAS 70895-01-1; Bromadol HCL; BDPC Hcl; 4-(4-bromophenyl)-4-(dimethylamino)-1-(2-phenylethyl)cyclohexanol; CAS 77239-98-6